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Brilanestrant (GDC-0810)

CAT: 0957-S7855Size: 5 mgDry Ice: YesHazardous: No
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CAT#:0957-S7855Size:5 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
Brilanestrant (GDC-0810, ARN-810) is a potent ER-α binder (ER-α, IC50 = 6.1 nM; ER-β, IC50 = 8.8 nM), a full transcriptional antagonist with no agonism and displays good potency and efficacy in ER-α degradation (EC50 = 0.7 nM) and MCF-7 breast cancer cell viability (IC50 = 2.5 nM) assays with good selectivity over other nuclear hormone receptors.
CAS Number
1365888-06-7
Synonyms
ARN-810
Target
Estrogen/progestogen Receptor
Activity
Endocrinology & Hormones
Molecular Formula
C26H20ClFN2O2
Storage Conditions
2 years -80 in solvent

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