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Rolapitant

CAT: 0957-S5476-01Size: 5 mgDry Ice: NoHazardous: No
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CAT#:0957-S5476-01Size:5 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
Rolapitant (SCH-619734) is a selective and competitive antagonist of human substance P/NK1 receptors with antiemetic activity. It has a high affinity for the human NK1 receptor of 0.66 nM and high selectivity over the human NK2 and NK3 subtypes of >1000-fold, as well as preferential affinity for human, guinea pig, gerbil and monkey NK1 receptors over rat, mouse and rabbit.
CAS Number
552292-08-7
Synonyms
SCH-619734
Target
Neurokinin Receptor
Activity
Neuronal Signaling
Molecular Formula
C25H26F6N2O2
Storage Conditions
3 years -20°C powder