Products for Research Use Only

GSK046 (iBET-BD2)

CAT: 0957-S9684-01Size: 5 mgDry Ice: NoHazardous: No
Product image 1
1 / 1
CAT#:0957-S9684-01Size:5 mg
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
Quick Request Actions
Description
GSK046 (iBET-BD2) is a selective and orally active inhibitor of BET (bromodomain and extraterminal domain) with IC50 of 264 nM, 98 nM, 49 nM and 214 nM for BRD2BD2, BRD3BD2, BRD4BD2 and BRDTBD2, respectively. GSK046 exhibits immunomodulatory activity.
CAS Number
2474876-09-8
Target
Epigenetic Reader Domain
Activity
Epigenetics
Molecular Formula
C23H27FN2O4
Storage Conditions
3 years -20°C powder