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KGA-2727

CAT: 0957-S8938-01Size: 5 mgDry Ice: NoHazardous: No
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CAT#:0957-S8938-01Size:5 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
KGA-2727 is a potent, selective, high-affinity inhibitor of sodium glucose cotransporter 1 (SGLT1) with Ki of 97.4 nM and 43.5 nM for human SGLT1 and rat SGLT1, respectively. The selectivity ratios (Ki for SGLT2/Ki for SGLT1) of KGA-2727 are 140 (human) and 390 (rat) . KGA-2727 exhibits antidiabetic efficacy in rodent models.
CAS Number
666842-36-0
Target
SGLT
Activity
GPCR & G Protein
Molecular Formula
C26H40N4O8
Storage Conditions
3 years -20°C powder