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MYCi361

CAT: 0957-S8905-01Size: 5 mgDry Ice: NoHazardous: No
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CAT#:0957-S8905-01Size:5 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
MYCi361 is a MYC inhibitor that engages MYC inside cells, disrupts MYC/MAX dimers, and impairs MYC-driven gene expression. MYCi361 binds to MYC with Kd of 3.2 μM. MYCi361 suppresses in vivo tumor growth, increases tumor immune cell infiltration, upregulates PD-L1 on tumors, and sensitizes tumors to anti-PD1 immunotherapy.
CAS Number
2289690-31-7
Synonyms
NUCC-0196361
Target
Myc
Activity
Apoptosis
Molecular Formula
C26H16ClF9N2O2
Storage Conditions
3 years -20°C powder