Products for Research Use Only

Pralsetinib (BLU-667)

CAT: 0957-S8716-01Size: 2 mgDry Ice: NoHazardous: No
Product image 1
1 / 1
CAT#:0957-S8716-01Size:2 mg
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
Quick Request Actions
Description
Pralsetinib (BLU-667, CS 3009, Gavreto) is a highly potent and selective RET (c-RET) inhibitor with an IC50 of 0.4 nM for WT RET. It also demonstrates potent activity (IC50 0.4 nmol/L) against common oncogenic RET alterations, including RET (M918T) .
CAS Number
2097132-94-8
Synonyms
CS 3009, Gavreto
Target
C-RET
Activity
Protein Tyrosine Kinase
Molecular Formula
C27H32FN9O2
Storage Conditions
3 years -20°C powder