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Avapritinib

CAT: 0957-S8553-01Size: 2 mgDry Ice: YesHazardous: No
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CAT#:0957-S8553-01Size:2 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
Avapritinib is a small molecule kinase inhibitor that potently inhibits PDGFRα D842V mutant activity in vitro (IC50 = 0.5 nM) and PDGFRα D842V autophosphorylation in the cellular setting (IC50 = 30 nM) ; also a potent inhibitor of the analogous Kit (c-Kit) mutation, D816V in Kit (c-Kit) Exon 17 (IC50 = 0.5 nM) .
CAS Number
1703793-34-3
Synonyms
BLU-285
Target
PDGFR
Activity
Protein Tyrosine Kinase
Molecular Formula
C26H27FN10
Storage Conditions
2 years -80 in solvent

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A19505-25Avapritinib 25mg
A19505-500Avapritinib 500mg
A19505-10Avapritinib 10mg
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