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TAK-243 (MLN7243)

CAT: 0957-S8341-01Size: 2 mgDry Ice: NoHazardous: No
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CAT#:0957-S8341-01Size:2 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
TAK-243 (MLN7243) is a potent, mechanism-based small-molecule inhibitor of the ubiquitin activating enzyme (UAE) with an IC50 of 1 ± 0.2 nM in the UBCH10 E2 thioester assay. It has minimal inhibitory activity in a panel of kinase and receptor assays, as well as on human carbonic anhydrase type I and type II. TAK-243 (MLN7243) induces ER stress, abrogates NFκB pathway activation and promotes apoptosis.
CAS Number
1450833-55-2
Target
E1 Activating
Activity
Ubiquitin
Molecular Formula
C19H20F3N5O5S2
Storage Conditions
3 years -20°C powder

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