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Salirasib

CAT: 0957-S7684-01Size: 5 mgDry Ice: YesHazardous: No
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CAT#:0957-S7684-01Size:5 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
Salirasib (Farnesylthiosalicylic acid, FTS) is a potent competitive prenylated protein methyltransferase (PPMTase) inhibitor with Ki of 2.6 μM, which inhibits Ras methylation. Salirasib exerts antitumor effects and induces autophagy. Phase 2.
CAS Number
162520-00-5
Synonyms
Farnesylthiosalicylic acid, FTS
Target
Ras
Activity
Apoptosis
Molecular Formula
C22H30O2S
Storage Conditions
2 years -80 in solvent