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Lestaurtinib

CAT: 0957-S7640Size: 5 mgDry Ice: NoHazardous: No
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CAT#:0957-S7640Size:5 mg
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Description
Lestaurtinib (CEP-701, KT-5555) is a derivative of the indolocarbazole K252 and a staurosporine analog. It is an orally active inhibitor of receptor protein tyrosine kinases (RPTKs), which inhibits FLT3 and Trk, with an IC50 of 3 nM and < 25 nM, respectively. It also inhibits JAK2 with an IC50 of 0.9 nM.
CAS Number
111358-88-4
Synonyms
CEP-701, KT-5555
Target
FLT3
Activity
Protein Tyrosine Kinase
Molecular Formula
C26H21N3O4

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