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WH-4-023

CAT: 0957-S7565-01Size: 5 mgDry Ice: YesHazardous: No
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CAT#:0957-S7565-01Size:5 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
WH-4-023 (KIN001-112, KIN112, Dual LCK/SRC inhibitor) is a potent and orally active Lck/Src inhibitor with IC50s of 2 nM and 6 nM in cell-free assays, respectively. Exhibits >300-fold selectivity against p38α and KDR. Also potently inhibits SIK (IC50 values are 10, 22 and 60 nM for SIK 1, 2 and 3 respectively) and displays selectivity over a range of closely related kinases.
CAS Number
837422-57-8
Synonyms
KIN001-112, KIN112, Dual LCK/SRC inhibitor
Target
Src
Activity
Protein Tyrosine Kinase
Molecular Formula
C32H36N6O4
Storage Conditions
2 years -80 in solvent

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