Products for Research Use Only

Epertinib hydrochloride

CAT: 0957-S6897-01Size: 5 mgDry Ice: NoHazardous: No
Product image 1
1 / 1
CAT#:0957-S6897-01Size:5 mg
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
Quick Request Actions
Description
Epertinib hydrochloride (S-222611 hydrochloride) is a potent, orally active, reversible, and selective tyrosine kinase inhibitor of EGFR, HER2 and HER4 with IC50 of 1.48 nM, 7.15 nM and 2.49 nM, respectively. Epertinib hydrochloride (S-222611 hydrochloride) exhibits antitumor activity.
CAS Number
2071195-74-7
Synonyms
Epertinib HCl, S-222611 hydrochloride, S-222611 HCl
Target
EGFR
Activity
Protein Tyrosine Kinase
Molecular Formula
C30H28Cl2FN5O3
Storage Conditions
3 years -20°C powder