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MK-2461

CAT: 0957-S2774Size: 5 mgDry Ice: YesHazardous: No
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CAT#:0957-S2774Size:5 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
MK-2461 is a potent, multi-targeted inhibitor for c-Met (WT/mutants) with IC50 of 0.4-2.5 nM, less potent to Ron, Flt1; 8- to 30-fold greater selectivity of c-Met targets versus FGFR1, FGFR2, FGFR3, PDGFRβ, KDR, Flt3, Flt4, TrkA, and TrkB. Phase 1/2.
CAS Number
917879-39-1
Target
C-Met
Activity
Protein Tyrosine Kinase
Molecular Formula
C24H25N5O5S
Storage Conditions
2 years -80 in solvent