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PF-04691502

CAT: 0957-S2743-01Size: 5 mgDry Ice: YesHazardous: No
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CAT#:0957-S2743-01Size:5 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
PF-04691502 (PF4691502) is an ATP-competitive PI3K (α/β/δ/γ) /mTOR dual inhibitor with Ki of 1.8 nM/2.1 nM/1.6 nM/1.9 nM and 16 nM in cell-free assays, little activity against either Vps34, AKT, PDK1, p70S6K, MEK, ERK, p38, or JNK. PF-04691502 induces apoptosis. Phase 2.
CAS Number
1013101-36-4
Synonyms
PF4691502
Target
Akt
Activity
PI3K/Akt/mTOR
Molecular Formula
C22H27N5O4
Storage Conditions
2 years -80 in solvent