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Niraparib (MK-4827)

CAT: 0957-S2741-01Size: 5 mgDry Ice: YesHazardous: No
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CAT#:0957-S2741-01Size:5 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
Niraparib (MK-4827) is a selective inhibitor of PARP1/2 with IC50 of 3.8 nM/2.1 nM, with great activity in cancer cells with mutant BRCA-1 and BRCA-2. It is >330-fold selective against PARP3, V-PARP and Tank1. Niraparib can form PARP–DNA complexes resulting in DNA damage, apoptosis, and cell death. Phase 3.
CAS Number
1038915-60-4
Target
PARP
Activity
DNA Damage/DNA Repair
Molecular Formula
C19H20N4O
Storage Conditions
2 years -80 in solvent

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