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Sapitinib (AZD8931)

CAT: 0957-S2192-01Size: 5 mgDry Ice: YesHazardous: No
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CAT#:0957-S2192-01Size:5 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
Sapitinib (AZD8931) is a reversible, ATP competitive inhibitor of EGFR, ErbB2 and ErbB3 with IC50 of 4 nM, 3 nM and 4 nM in cell-free assays, more potent against NSCLC cell, 100-fold more selective for the ErbB family than MNK1 and Flt. Phase 2.
CAS Number
848942-61-0
Target
EGFR
Activity
Protein Tyrosine Kinase
Molecular Formula
C23H25ClFN5O3
Storage Conditions
2 years -80 in solvent