Products for Research Use Only

BGB-3245 (Brimarafenib)

CAT: 0957-E4599-01Size: 1 mgDry Ice: NoHazardous: No
Product image 1
1 / 1
CAT#:0957-E4599-01Size:1 mg
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
Quick Request Actions
Description
BGB-3245 (Brimarafenib, Brimarafenibum) is an inhibitor of Raf kinase. BGB-3245 displays potent effects against different RAF isoforms, including BRAF Class I/II/III mutations, BRAF fusions, and heterodimerization with CRAF in preclinical models. It also exhibits antineoplastic effects.
CAS Number
1643326-82-2
Synonyms
Brimarafenib, Brimarafenibum
Target
Raf
Activity
MAPK
Molecular Formula
C24H17F3N4O4