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M2912

CAT: 0957-E1069-01Size: 5 mgDry Ice: NoHazardous: No
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CAT#:0957-E1069-01Size:5 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
M2912 (MSC2504877) is a very potent TNKS1/TNKS2 inhibitor (IC50=0.6 nM for TNKS1) with exquisite selectivity over other PARP family enzymes and favorable compound properties. This inhibitor potently modulates the Wnt/β-catenin pathway by elevating the levels of axin2 (EC50=17 nM) and tankyrase in DLD1 cells in a dose-dependent manner resulting in reduced cellular Wnt reporter activity.
CAS Number
1460286-21-8
Synonyms
MSC2504877
Target
PARP
Activity
DNA Damage/DNA Repair
Molecular Formula
C17H18N2O2
Storage Conditions
3 years -20°C powder

Alternative Products

CatalogName
C01460-5mgM2912

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