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GNE-781

CAT: 0957-S8665-01Size: 5 mgDry Ice: NoHazardous: No
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CAT#:0957-S8665-01Size:5 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
GNE-781 (compound 19) is an orally active, highly potent and selective bromodomain inhibitor of cyclic adenosine monophosphate response element binding protein (CBP) with IC50 of 0.94 nM in TR-FRET assay. GNE-781 also inhibits BRET and BRD4 (1) with IC50 of 6.2 nM and 5100 nM, respectively. GNE-781 exhibits antitumor activity.
CAS Number
1936422-33-1
Target
Epigenetic Reader Domain
Activity
Epigenetics
Molecular Formula
C27H33F2N7O2
Storage Conditions
3 years -20°C powder

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