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PF-06726304

CAT: 0957-S8494-01Size: 2 mgDry Ice: YesHazardous: No
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CAT#:0957-S8494-01Size:2 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
PF-06726304 is a selective EZH2 inhibitor with Ki values of 0.7 nM and 3 nM for WT EZH2 and Y641N respectively; also inhibits H3K27me3 with the IC50 value of 15 nM.
CAS Number
1616287-82-1
Synonyms
PF-6726304
Target
Histone Methyltransferase
Activity
Epigenetics
Molecular Formula
C22H21Cl2N3O3
Storage Conditions
2 years -80 in solvent