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Alvelestat (AZD9668)

CAT: 0957-S7218-01Size: 5 mgDry Ice: YesHazardous: No
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CAT#:0957-S7218-01Size:5 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
Alvelestat (AZD9668, Avelestat) is an oral, highly selective inhibitor of neutrophil elastase (NE) with IC50 and Ki of 12 nM and 9.4 nM, at least 600-fold more selective over other serine proteases. Phase 2.
CAS Number
848141-11-7
Synonyms
Avelestat
Target
Serine Protease
Activity
Proteases
Molecular Formula
C25H22F3N5O4S
Storage Conditions
2 years -80 in solvent

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