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Lonafarnib (SCH66336)

CAT: 0957-S2797-01Size: 5 mgDry Ice: YesHazardous: No
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CAT#:0957-S2797-01Size:5 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
Lonafarnib (SCH66336) is an orally bioavailable FPTase inhibitor for H-ras, K-ras-4B and N-ras with IC50 of 1.9 nM, 5.2 nM and 2.8 nM in cell-free assays, respectively. Phase 3.
CAS Number
193275-84-2
Target
Transferase
Activity
Metabolism
Molecular Formula
C27H31Br2ClN4O2
Storage Conditions
2 years -80 in solvent