Atazanavir

CAT: 0498-bs-83448C-01Size: 10 mgDry Ice: NoHazardous: No
CAT#:0498-bs-83448C-01Size:10 mg
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AVAILABILITY: InStock
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Background
An azapeptide-based inhibitor of HIV protease (Ki = 2.66 nM) .1 Inhibits SARS-CoV-2 main protease (Ki = 703 nM), but not papain-like protease (Ki = 9.87 µM) .2 Blocks SARS-CoV-2 replication and IL-6 / TNFα production in vitro.3 Also inhibits the liver enzyme UDP-glucuronyltransferase 1A1 (UGT1A1), IC50 = 160 nM for recombinant UGT1A1.4
Conjugation
Unconjugated
Buffer
White to off-white solid
Storage Conditions
-20°C

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