Products for Research Use Only

Luminespib

CAT: 0498-bs-82980C-01Size: 5 mgDry Ice: NoHazardous: No
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CAT#:0498-bs-82980C-01Size:5 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Background
Luminespib is a potent inhibitor (IC50 = 21 nM) of HSP90.1 It is active against various human tumor xenograft models acting via several processes including cytostasis, apoptosis, invasion, and angiogenesis.2,3 Luminespib enhances tumor susceptibility to T-cell-based immunotherapy by re-invigorating the cancer-immunity cycle in NANOG+ cancer cells.4 It also acts as a radiosensitizer against various tumor cells.5-7
Conjugation
Unconjugated
Buffer
White solid
Storage Conditions
-20°C