R 892

• Description :

  Potent and selective bradykinin B1 receptor antagonist (ID50 values are 2.8 and > 600 nM at B1 and B2 receptors respectively) . Exhibits no intrinsic agonist activity and is resistant to aminopeptidase and kininase II (ACE) cleavage. Displays hypertensive activity in vivo.

• Stability :

  ≥ 2 years

• Purity :

  >98% (HPLC)

• Weight :

  1154.37

• Molecular Formula :

  C58H83N13O12

• Notes :

  Research use only, not for human use.

• Receptor :

  ——

• CAS Number :

  229030-05-1