JKC 363

• Description :

  Potent and selective melanocortin MC4 receptor antagonist (IC50 values are 0.5 and 44.9 nM at MC4 and MC3 respectively) that antagonizes the effects of α-MSH. Suppresses thyrotropin-releasing hormone (TRH) release, attenuates food intake and reduces formalin-induced pain in vivo.

• CAS Number :

  436083-30-6

• Stability :

  ≥ 2 years

• Purity :

  >98% (HPLC)

• Weight :

  1506.72

• Molecular Formula :

  C69H91N19O16S2

• Notes :

  Research use only, not for human use.

• Receptor :

  ——