MSG 606

• Description :

  Potent human MC1 receptor antagonist (IC50 = 17 nM) . Also partial agonist at human MC3 and MC5 receptors (EC50 values are 59 and 1300 nM, respectively) . Exhibits binding affinity for A375 melanoma cells in vitro. Reverses morphine-induced hyperalgesia in female mice, with no effect in male mice. γMSH analog.

• Stability :

  ≥ 2 years

• Purity :

  >98% (HPLC)

• Weight :

  1347.51

• Molecular Formula :

  C62H82N20O13S

• Notes :

  Research use only, not for human use.

• Receptor :

  ——

• CAS Number :

  1416983-77-1