MEN 11270

• Description :

  Peptide antagonist of the B2 bradykinin receptor (pKi = 10.3) ; conformationally constrained cyclized analog of HOE 140. Blocks hypotension and bronchoconstriction in vivo. Displays selectivity for B2 over 29 other receptors and ion channels (pIC50 < 5.5) .

• Stability :

  ≥ 2 years

• Purity :

  >98% (HPLC)

• Weight :

  1299.56

• Molecular Formula :

  C60H90N20O11S

• Notes :

  Research use only, not for human use.

• Receptor :

  ——

• CAS Number :

  235082-52-7