PKC β pseudosubstrate

• Description :

  Selective cell-permeable peptide inhibitor of protein kinase C (IC50 ~ 0.5 μM) . Consists of amino acids 19 - 31 of PKC pseudosubstrate domain linked by a disulphide bridge to a cell permeabilisation Antennapedia domain vector peptide. The Antennapedia peptide is actively taken up by intact cells, at 4 or 37°C, ensuring rapid and effective uptake of the inhibitor peptide. Once inside the cell, the disulphide bonds are subjected to reduction in the cytoplasm leading to release of the inhibitor peptide.

• Stability :

  ≥ 2 years

• Purity :

  >98% (HPLC)

• Weight :

  3994.84

• Molecular Formula :

  C177H294N62O38S3

• Notes :

  Research use only, not for human use.

• Receptor :

  ——

• CAS Number :

  172308-76-8