APETx2

• Description:

  Acid-sensing ion channel 3 (ASIC3) channel blocker (IC50 values are 63 and 175 nM for homomeric rat and human ASIC3 channels) . Also inhibits NaV1.8 and NaV1.2 channels (IC50 values are 55 and 114 nM respectively) . Demonstrates analgesic properties against acid-induced and inflammatory pain.

• Stability:

  ≥ 2 years

• Purity:

  >98% (HPLC)

• Weight:

  4561.06

• Molecular Formula:

  C196H280N54O61S6

• Notes:

  Research use only, not for human use.

• Receptor:

  ——

• CAS Number:

  713544-47-9