WDR5-0102

• Description:

  WDR5-0102 is a compound that inhibits the WDR5-MLL1 interface (K dis = 7 μM, K d = 4 μM), selectively reducing MLL1 HMT activity without affecting the human H3K4 methyltransferase SETD7 or other HMTs, including G9a, EHMT1, SUV39H2, SETD8, PRMT3, and PRMT5.

• Stability:

  ≥ 2 years

• Purity:

  >98% (HPLC)

• Weight:

  374.82

• Molecular Formula:

  C18H19ClN4O3

• Notes:

  Research use only, not for human use.

• Receptor:

  Histone Methyltransferase

• CAS Number:

  824960-50-1