Mardepodect hydrochloride

• Description:

  Mardepodect hydrochloride (Mardepodect HCl) is an orally active, selective and potent inhibitor of PDE10A that crosses the blood-brain barrier (IC50: 0.37 nM) .Mardepodect hydrochloride up-regulates the expression of proteins encoding specific growth and transcription factors, cell signalling molecules and cell surface proteins. Mardepodect hydrochloride upregulates genes encoding specific growth factors, transcription factors, cell signalling molecules, and cell surface proteins, while downregulating a broad spectrum of cell cycle and apoptosis-related genes.

• Stability:

  ≥ 2 years

• Purity:

  >98% (HPLC)

• Weight:

  428.91

• Molecular Formula:

  C25H21ClN4O

• Notes:

  Research use only, not for human use.

• Receptor:

  Apoptosis | PDE

• CAS Number:

  2070014-78-5