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PBRM1-BD2-IN-5

CAT: 1410-M35352-01Size: 1 mL x 10 mM in DMSODry Ice: NoHazardous: No
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CAT#:1410-M35352-01Size:1 mL x 10 mM in DMSO
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
PBRM1-BD2-IN-5 is a potent inhibitor of the PBRM1 Bromodomain, with dissociation constant (Kd) values of 1.5 μM and 3.9 μM for PBRM1-BD2 and PBRM1-BD5 respectively, and an inhibitory concentration 50 (IC50) value of 0.26 μM for PBRM1-BD2. This compound effectively diminishes the interaction between full-length PBRM1 and acetylated histone peptide within the PBAF complex in cell lysates, making it a promising candidate for anticancer research.
CAS Number
2819989-61-0
Stability
≥ 2 years
Purity
>98% (HPLC)
Weight
272.73
Molecular Formula
C15H13ClN2O
Notes
Research use only, not for human use.
Receptor
Epigenetic Reader Domain

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