GP 1a

• Description:

  GP 1a is a potent agonist of cannabinoid receptor 2 (CB2) (EC50=7.1), as shown in cAMP, GTPγS and β-arrestin recruitment assays. GP 1a is approximately 30-fold more selective for CB2 receptors than CB1 receptors and increases P-ERK1/2 expression in HL-60 cells in vitro. GP 1a is beneficial for skin wound healing. GP 1a inhibits inflammation and fibrogenesis while promoting epithelial re-formation.

• Stability:

  ≥ 2 years

• Purity:

  >98% (HPLC)

• Weight:

  441.35

• Molecular Formula:

  C23H22Cl2N4O

• Notes:

  Research use only, not for human use.

• Receptor:

  Cannabinoid Receptor | PERK

• CAS Number:

  511532-96-0