ZEN-3219

• Description:

  ZEN-3219 is a BET inhibitor, which has inhibitory effect on BRD4 (BD1), BRD4 (BD2) and BRD4 (BD1BD2) . ZEN-3219 has inhibitory effect on BRD4 (BD1), The IC50 values of BRD4 (BD2) and BRD4 (BD1BD2) were 0.48, 0.16 and 0.47 μM, respectively. ZEN-3219 is a component of PROTAC molecule and can induce BRD4 degradation.

• Stability:

  ≥ 2 years

• Purity:

  >98% (HPLC)

• Weight:

  322.36

• Molecular Formula:

  C19H18N2O3

• Notes:

  Research use only, not for human use.

• Receptor:

  Epigenetic Reader Domain

• CAS Number:

  1952264-34-4