Products for Research Use Only

GSK778

CAT: 1410-M28843-01Size: 1 mL x 10 mM in DMSODry Ice: NoHazardous: No
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CAT#:1410-M28843-01Size:1 mL x 10 mM in DMSO
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
GSK778 is a potent and selective inhibitor of BD1 bromodomain such as BRD2 BD1 (IC50s = 75 nM), BRD3 BD1 (IC50s = 41 nM), BRD4 BD1 (IC50s = 41 nM), and BRDT BD1 (IC50s = 143 nM) . GSK778 inhibits proliferation, induces a cell cycle arrest and apoptosis.
CAS Number
2451862-42-1
Stability
≥ 2 years
Purity
>98% (HPLC)
Weight
511.61
Molecular Formula
C30H33N5O3
Notes
Research use only, not for human use.
Receptor
VHL