BMS-986122

• Description:

  BMS 986122 is a positive allosteric modulator of μ-opioid receptors that increases β-arrestin recruitment stimulated by endomorphin 1 in U2OS-OPRM1 human osteosarcoma cells expressing μ-opioid receptors (EC50 = 3 μM) .

• Stability:

  ≥ 2 years

• Purity:

  >98% (HPLC)

• Weight:

  448.77

• Molecular Formula:

  C16H15BrClNO3S2

• Notes:

  Research use only, not for human use.

• Receptor:

  FAP

• CAS Number:

  313669-88-4