MDR-652

• Description :

  MDR-652 is a highly specific and efficacious agonist of nonpungent transient receptor potential vanilloid 1 (TRPV1) with Ki value of 11.4 nM and 23.8 nM for hTRPV1 and rTRPV1 respectively and EC50s for hTRPV1 and rTRPV1 are 5.05 and 93 nM respectively.

• Stability :

  ≥ 2 years

• Purity :

  >98% (HPLC)

• Weight :

  447.95

• Molecular Formula :

  C22H23ClFN3O2S

• Notes :

  Research use only, not for human use.

• Receptor :

  BET bromodomain|Apoptosis|BRD2|BRD3|BRD4

• CAS Number :

  1933528-96-1