BSJ-4-116

• Description :

  BSJ-4-116 is a highly potent and selective CDK12 degrader (PROTAC) with an IC50 of 6 nM. It downregulates DDR genes through a premature termination of transcription, primarily through increasing poly (adenylation) .

• Stability :

  ≥ 2 years

• Purity :

  >98% (HPLC)

• Weight :

  837.38

• Molecular Formula :

  C40H49ClN8O8S

• Notes :

  Research use only, not for human use.

• Receptor :

  CDK12|Cereblon

• CAS Number :

  2519823-34-6