AM095 free acid

• Description:

  AM095 (free acid) is a potent LPA1 receptor antagonist (IC50s: 0.98 and 0.73 μM for recombinant human or mouse LPA1) .In vitro, AM095 was a potent LPA receptor antagonist because it inhibited GTPγS binding to Chinese hamster ovary (CHO) cell membranes overexpressing recombinant human or mouse LPA with IC values of 0.98 and 0.73 μM, respectively, and exhibited no LPA agonism.

• Stability:

  ≥ 2 years

• Purity:

  >98% (HPLC)

• Weight:

  456.49

• Molecular Formula:

  C27H24N2O5

• Notes:

  Research use only, not for human use.

• Receptor:

  LPA1

• CAS Number:

  1228690-36-5