PRX-07034

• Description:

  PRX-07034 is a selective antagonist of 5-HT6 receptor. It has cognition and memory-enhancing properties and potently decreases food intake and body weight in rodents. PRX-07034 is both a potent (Ki = 4-8 nM) and highly selective 5-HT (6) receptor antagonist (≥100-fold selectivity for the 5-HT (6) receptor compared to 68 other GPCRs, ion channels, and transporters, except D (3) (Ki = 71 nM) and 5-HT (1B) (Ki = 260 nM) receptors.

• Stability:

  ≥ 2 years

• Purity:

  >98% (HPLC)

• Weight:

  490.44

• Molecular Formula:

  C21H29Cl2N3O4S

• Notes:

  Research use only, not for human use.

• Receptor:

  5-HT6

• CAS Number:

  903580-39-2