MM-102 TFA

• Description:

  MM-102 TFA is a potent WDR5/MLL interaction inhibitor, achieves IC50 = 2.4 nM. MM-102 compound prevents the interaction between mixed lineage leukemia 1 (MLL1) and WD Trp-Asp repeat domain 5 (WDR5) and results in the inhibition of MLL1 H3K4 histone methyltransferase (HMT) activity.

• Stability:

  ≥ 2 years

• Purity:

  >98% (HPLC)

• Weight:

  783.83

• Molecular Formula:

  C37H50F5N7O6

• Notes:

  Research use only, not for human use.

• Receptor:

  MLL1

• CAS Number:

  1883545-52-5