PKR-IN-C16

• Description:

  PKR-IN-C16 is a specific protein kinase (PKR) inhibitor. PKR-IN-C16 is able to inhibit the autophosphorylation of PKR and unlock the translation blockade induced by PKR in primary neuronal cultures.PKR-IN-C16 binds the ATP-binding site of PKR and blocks autophosphorylation with an IC50 value of 186-210 nM.

• Stability:

  ≥ 2 years

• Purity:

  >98% (HPLC)

• Weight:

  268.29

• Molecular Formula:

  C13H8N4OS

• Notes:

  Research use only, not for human use.

• Receptor:

  PKR

• CAS Number:

  608512-97-6