EGFR-IN-7

• Description:

  EGFR-IN-7 is a selective and potent EGFR kinase inhibitor.TQB3804 displayed potent enzymatic activities for EGFRd746-750/T790M/C797S, EGFRL858R/T790M/C797S, EGFRd746-750/T790M, and EGFRL858R/T790M with IC50 of 0.46, 0.13, 0.26, and 0.19 nM respectively, and has similar enzymatic activity for EGFRWT (IC50 = 1.07) to Osimertinib.

• Stability:

  ≥ 2 years

• Purity:

  >98% (HPLC)

• Weight:

  694.6

• Molecular Formula:

  C32H41BrN9O2P

• Notes:

  Research use only, not for human use.

• Receptor:

  EGFR

• CAS Number:

  2267329-76-8