Otenabant

• Description:

  A potent, and selective CB1 receptor antagonist with Ki of 0.7 nM/0.12 nM in binding and functional assays respectively; has low affinity (Ki=7600 nM) for human CB2 receptors; reverses cannabinoid agonist mediated responses, reduces food intake, and increases energy expenditure and fat oxidation in rodents.ObesityPhase 3 Discontinued

• Stability:

  ≥ 2 years

• Purity:

  >98% (HPLC)

• Weight:

  510.4183

• Molecular Formula:

  C25H25Cl2N7O

• Notes:

  Research use only, not for human use.

• Receptor:

  CB1

• CAS Number:

  686344-29-6