LY-364947

• Description:

  LY364947 is a potent ATP-competitive inhibitor of TGFβR-I with IC50 of 59 nM in a cell-free assay, shows 7-fold selectivity over TGFβR-II.

• Stability:

  ≥ 2 years

• Purity:

  >98% (HPLC)

• Weight:

  272.3

• Molecular Formula:

  C17H12N4

• Notes:

  Research use only, not for human use.

• Receptor:

  CK1δ| MLK-7K| TGFβRI| TGFβRII| RIPK2

• CAS Number:

  396129-53-6