Rislenemdaz mesylate

CAT:
1410-M12971-01
Size:
1 g
  • Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
  • Dry Ice Shipment: No
Rislenemdaz mesylate - image 1

Rislenemdaz mesylate

  • Description:

    Rislenemdaz (MK 0657; CERC 301) is a potent, orally bioavailable, brain‐penetrant, NR2B-selective NMDA receptor (GluN2B) antagonist with Ki and IC 50 of 8.1 nM and 3.6 nM respectively.
  • Stability:

    ≥ 2 years
  • Purity:

    >98% (HPLC)
  • Weight:

    454.517
  • Molecular Formula:

    C20H27FN4O5S
  • Notes:

    Research use only, not for human use.
  • Receptor:

    IGluR
  • CAS Number:

    1893392-76-1