THIQ 40

• Description:

  THIQ 40 (THIQ40) is a potent, orally available ERα antagonist and selective estrogen receptor degrader (SERD) with IC50 of 17 nM (ERα binding) and 30 nM (ERα transcription), IC50 of 0.9 nM (ERα degradation) .

• Stability:

  ≥ 2 years

• Purity:

  >98% (HPLC)

• Weight:

  427.544

• Molecular Formula:

  C28H29NO3

• Notes:

  Research use only, not for human use.

• Receptor:

  Estrogen Receptor/ERR

• CAS Number:

  1799430-91-3