PF-05190457

• Description:

  A potent, selective, and orally bioavailable ghrelin receptor (GHSR) inverse agonist with binding pKi of 8.36; displays excellent off-target activity in the CEREP panel at 10 uM with exception of serotonin 5-HT2B (IC50=3.7 uM) .

• Stability:

  ≥ 2 years

• Purity:

  >98% (HPLC)

• Weight:

  512.676

• Molecular Formula:

  C29H32N6OS

• Notes:

  Research use only, not for human use.

• Receptor:

  GHSR

• CAS Number:

  1334782-79-4