Products for Research Use Only

FMJ-01-054

CAT: 0013-GTR19274800-01Size: 10 mgDry Ice: NoHazardous: No
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CAT#:0013-GTR19274800-01Size:10 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
FMJ-01-054 is a selective dopamine D4 receptor (D4R) antagonist with a Ki value of 77.7 nM. It exhibits subtype selectivity for D2R and D3R. FMJ-01-054 inhibits D4R-mediated β-arrestin recruitment and cAMP production, with IC50 values of 3800 nM and 134 nM, respectively. In rats, it demonstrates an ideal plasma half-life and brain exposure. FMJ-01-054 is applicable in neuropsychiatric disorder research.
Storage Conditions
-20°C
Notes
For research use only.

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